New explortion of 1,1-Dioxo-isothiazolidine

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Chemistry is an experimental science, and the best way to enjoy it and learn about it is performing experiments. 5908-62-3. Introducing a new discovery about 5908-62-3, Name is 1,1-Dioxo-isothiazolidine

Discovery of potent HIV integrase inhibitors active against raltegravir resistant viruses

A series of novel HIV integrase inhibitors active against rategravir resistant strains are reported. Initial SAR studies revealed that activities against wild-type virus were successfully maintained at single digit nanomolar level with a wide range of substitutions. However, inclusion of nitrogen-based cyclic substitutions was crucial for achieving potency against mutant viruses. Several compounds with excellent activities against wild-type virus as well as against the viruses with the mutations Q148H/G140S or N155H/E92Q were reported.

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Reference£º
Quinuclidine – Wikipedia,
Quinuclidine | C7H578N | ChemSpider